Moetsi oa phofo ea Galantamine Hydrobromide Nomoro ea CAS: 1953-04-4 Bohloeki ba 98% bonyane bakeng sa metsoako ea tlatsetso
Liparamente tsa Sehlahisoa
| Lebitso la sehlahisoa | Galantamine Hydrobromide |
| Lebitso le leng | Galanthamine hydrobromide; Galantamine HBr; Galanthamine HBr;(4aS,6R,8aS)-4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef][2]benzazepin-6-ol, Hydrobromide |
| Nomoro ea CAS | 1953-04-4 |
| Foromo ea limolek'hule | C17H21NO3.HBr |
| Boima ba limolek'hule | 368.27 |
| Bohloeki | 98.0% |
| Ponahalo | phofo e tšoeu ho isa ho e tšoeu |
| Ho paka | 1kg/mokotla 10kgs ,25kgs/moropa |
| Kopo | lithethefatsi tsa nootropic |
Selelekela sa sehlahisoa
Galantamine hydrobromide ke benzazepine e nkiloeng ho tsoa li-bulbs le lipalesa tsa narcissus, osmanthus, kapa canna. Hape ke thibelo ea cholinesterase ea molomo. E le ligand bakeng sa li-receptor tsa nicotinic acetylcholine, e 'nile ea sebelisoa haholo ho ntlafatsa ts'ebetso ea methapo ea kutlo. Mosebetsi oa eona ke ho thibela acetylcholinesterase ka tlholisano le ka mokhoa o khutlisetsang morao, ka hona e eketsa khatello ea acetylcholine. Ha e monngoa maling, galantamine hydrobromide e monngoa habonolo likarolong tse fapaneng tsa' mele, ho kenyeletsoa le boko. E tlama ho li-receptor tsa nicotinic acetylcholine, e baka liphetoho tsa sebopeho le ho eketsa ho lokolloa ha acetylcholine. E boetse e sebetsa ka ho qothisana lehlokoa le ho fetola litlamorao tsa li-inhibitor tsa cholinesterase. Ka ho thibela cholinesterase, e thibela ho senyeha ha acetylcholine, ka hona e eketsa maemo le nako ea neurotransmitter ena e matla. Galantamine e ka boela ea ntlafatsa ho ithuta le ho hopola, ea thibela ho ruruha ha boko, 'me ea boloka maemo a holimo a li-neurotransmitter ka ho boloka botšepehi ba li-neuron le li-synapses.
Tšobotsi
(1) Bohloeki bo phahameng: Galantamine hydrobromide e ka ba sehlahisoa se hloekileng haholo ka mekhoa ea tlhahiso ea ho hloekisa. Bohloeki bo phahameng bo bolela ho fumaneha habonolo ha 'mele le ho fokotsa likarabelo tse mpe.
(2) Polokeho: Galantamine hydrobromide e pakiloe e bolokehile bakeng sa 'mele oa motho.
(3) Botsitso: Galantamine hydrobromide e na le botsitso bo botle mme e ka boloka ts'ebetso le phello ea eona tlas'a maemo a fapaneng le maemo a polokelo.
Likopo
Jwalo ka tlatsetso ya dijo, galantamine hydrobromide e ka ntlafatsa mohopolo, temoho le bokgoni ba ho etsa mesebetsi ya letsatsi le letsatsi. E sebetsa ka ho tsosolosa tekano ya dintho tse itseng tsa tlhaho (di-neurotransmitters) bokong, e leng se eketsang lebelo la ho thehwa ha mohopolo le ho ntlafatsa ho boloka dintlha le dintlha. Ho feta moo, galantamine hydrobromide e ama neuroplasticity ka kotloloho kapa ka tsela e sa tobang. E hlasimolla synaptic plasticity ka ho kenya tshebetsong microglia le astrocytes. Galantamine e fana ka tshireletso ya antioxidant kgahlanong le kgatello ya oxidative e bakwang ke di-free radicals.












