PRL-8-53 moetsi oa phofo CAS No.: 51352-87-5 98% bohloeki min. bakeng sa lisebelisoa tsa tlatsetso
Lihlahisoa tsa lihlahisoa
| Lebitso la sehlahisoa | PRL-8-53 |
| Lebitso le leng | Methyl 3-(2-(benzyl(Methyl)aMino)ethyl)benzoate hydrochloride;Benzoic acid, 3-[2-[methyl(phenylmethyl)amino]ethyl]-, methyl ester, hydrochloride (1:1);Methyl 3- {2- [benzyl(methyl)amino]ethyl}benzoate hydrochloride (1:1) |
| Nomoro ea CAS. | 51352-87-5 |
| Mokhoa oa limolek'hule | C18H22ClNO2 |
| Boima ba molek'hule | 319.83 |
| Bohloeki | 98.0% |
| Ponahalo | Phofo e tšoeu |
| Ho paka | 1 kg ka mokotla 25kg / moropa |
| Kopo | nootropic |
Kenyelletso ea sehlahisoa
PRL-8-53, eo hape e tsejoang e le methyl 3- (2- (benzyl(methyl) amino) ethyl) benzoate, ke motsoako oa nootropic oa maiketsetso o nahanoang ho ntlafatsa phetiso ea cholinergic le ho laola maemo a dopamine bokong. Boitšoaro bona bo kenya letsoho litlamoraong tsa eona tse ka ntlafatsang mohopolo, ka hona, ho ntlafatsa sebopeho sa mohopolo, ho boloka, le ho khutlisa. Liphuputso tse ngata tse mabapi le liphoofolo le batho li tlalehile liphello tse ntle bakeng sa thepa ea eona e ntlafatsang mohopolo. Phuputsong ea lifofane tse sa boneng habeli, tse laoloang ke placebo, batho ba fumaneng tekanyo e le 'ngoe ea PRL-8-53 ba bontšitse mohopolo o betere oa mantsoe le bokhoni ba ho khutlisa ha bo bapisoa le sehlopha sa placebo. Liphuputso tsena li ile tsa tsosa thahasello le lipatlisiso tse eketsehileng mabapi le bokhoni ba motsoako. Phuputso e 'ngoe ho likhoto e bontšitse hore ho fana ka PRL-8-53 ho ntlafalitse haholo bokhoni ba bona ba ho ithuta ka mosebetsi oa maze oa metsi. Likhoto tse tšoaroang ka PRL-8-53 li khonne ho fumana sethala se patiloeng ka mokhoa o atlehileng ho feta taolo, ho bonts'a bokhoni ba komporo joalo ka mohopolo o matlafatsang.
Sebopeho
(1) Bohloeki bo phahameng: PRL-8-53 e ka fumana lihlahisoa tse hloekileng ka ho hloekisa mekhoa ea tlhahiso. Bohloeki bo phahameng bo bolela bioavailability e betere le ho fokotseha ho hoholo ha maikutlo.
(2) Tšireletseho: Tšireletseho e phahameng, liketso tse fokolang tse fokolang, ha ho na liketso tse mpe tse totobetseng.
(3) Botsitso: PRL-8-53 e na le botsitso bo botle 'me e ka boloka ts'ebetso ea eona le phello tlas'a maemo a fapaneng le maemo a polokelo.
Lisebelisoa
E le mofuta o mocha oa tlatsetso ea ntlafatso ea kelello, PRL-8-53 e ntlafatsa mohopolo oa nako e khuts'oane le mohopolo o sebetsang, ha e ntse e ntlafatsa bokhoni ba ho ithuta le lebelo la ho fumana bokhoni, e thusa ho ntlafatsa ho ithuta le katleho ea mosebetsi. Lipatlisiso li bontša hore PRL-8-53 e ka khothalletsa kholo le tsosoloso ea li-neurone bokong. PRL-8-53 e ka eketsa lebelo leo boko bo sebetsanang le boitsebiso ka lona, ho lumella batho ho phetha mesebetsi le ho etsa liqeto kapele. Le hoja ho bapisoa le metsoako e meng ea nootropic Leha ho le joalo, lipatlisiso tsa PRL-8-53 li lekane, empa lipatlisiso tse teng li fana ka maikutlo a bokhoni ba eona ba ho ntlafatsa mohopolo le bokhoni ba kelello.
