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sehlahisoa

Tianeptine Semisulfate Monohydrate moetsi oa phofo CAS No.: 1224690-84-9 98% bohloeki min.bakeng sa lisebelisoa tsa tlatsetso

Tlhaloso e Khutšoanyane:

Tianeptine Hemisulfate Monohydrate ke serotonin reuptake inhibitor (SSRI) e khethiloeng le sethethefatsi se thibelang ho imeloa kelellong.


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Lihlahisoa tsa lihlahisoa

Lebitso la sehlahisoa

Tianeptine Hemisulfate Monohydrate

Lebitso le leng

tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2);

Tianeptinehemisulfatemonohydrate(THM);

7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2);

Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;

THM

Nomoro ea CAS.

1224690-84-9

Mokhoa oa limolek'hule

C21H27ClN2O8S2

Boima ba molek'hule

535.02

Bohloeki

98.0%

Ponahalo

Phofo e tšoeu ea kristale

Kopo

Tlatsetso ea Lijo tse tala

Kenyelletso ea sehlahisoa

Tianeptine Hemisulfate Monohydrate ke serotonin reuptake inhibitor (SSRI) e khethiloeng le sethethefatsi se thibelang ho imeloa kelellong.Joaloka moriana o sa tloaelehang oa ho tepella maikutlo, mokhoa oa eona oa ts'ebetso o fapane le oa li-antidepressants tsa setso, ho ntlafatsa maikutlo le boemo ba maikutlo ka ho matlafatsa synaptic plasticity ea hippocampal neurons.Tianeptine Hemisulfate Monohydrate e boetse e sebelisetsoa ho tšoara matšoenyeho le mathata a maikutlo.

Tianeptine Hemisulfate Monohydrate e sebelisoa haholo lipatlisisong tsa bongaka, haholo-holo ho nts'etsopele ea li-antidepressants.E ntse e etsoa lipatlisiso bakeng sa tšebeliso ea mafu a neurodegenerative, taolo ea bohloko, le kalafo ea bokhoba.Ts'ebetso ea Tianeptine Hemisulfate Monohydrate e 'nile ea ithutoa haholo' me ea tiisoa, 'me e amohetsoe bakeng sa phekolo ea ho tepella maikutlong linaheng tse ngata.

Hoa lokela ho hlokomeloa hore le hoja Tianeptine Hemisulfate Monohydrate e 'nile ea pakoa e le moriana o thibelang ho imeloa kelellong ka katleho lits'ebetsong tsa meriana, e khetholloa e le ntho e laoloang linaheng tse ling, e nang le lithibelo mabapi le tšebeliso ea eona le thekiso.Mang kapa mang ea sebelisang kapa a rekang Tianeptine Hemisulfate Monohydrate o lokela ho tseba melao le melaoana e amehang naheng ea habo bona.

Sebopeho

(1) Mokhoa o ikhethileng oa ts'ebetso: Tianeptine Hemisulfate Monohydrate ke serotonin reuptake enhancer (SSRE) e khethiloeng, e bolelang hore e ntlafatsa ho tsosolosoa ha serotonin bokong, e leng se lebisang ho eketseha ha polasetiki ea synaptic le ntlafatso ea maikutlo.Mokhoa ona oa ts'ebetso o fapane le li-antidepressants tsa setso, tseo hangata e leng serotonin reuptake inhibitors (SSRIs).
(2) Ts'ebetso e potlakileng ea ketso: Tianeptine Hemisulfate Monohydrate e na le ts'ebetso e potlakileng ea ts'ebetso, ka lithuto tsa kliniki tse bontšang ntlafatso ea matšoao a tepeletseng pele beke e le 'ngoe ka mor'a ho qala kalafo.
(3) Ts'ebetso e ntlafetseng ea ts'ebetso: Tianeptine Hemisulfate Monohydrate e bontšitsoe ho ntlafatsa ts'ebetso ea kelello ho bakuli ba nang le bothata bo boholo ba ho tepella maikutlo, joalo ka mohopolo le tlhokomelo.

(4) Bokhoni bo fokolang ba ho lemalla: Ho fapana le li-antidepressants tse ling, Tianeptine Hemisulfate Monohydrate e na le matla a fokolang a ho lemalla 'me ha e bake matšoao a ho ikhula ha e khaotsa.Lebaka ke hobane ha e shebane le sistimi ea dopamine, e amanang le bokhoba le boits'oaro.

(5) Kalafo ea mathata a ho tšoenyeha: Tianeptine Hemisulfate Monohydrate e bontšitsoe hore e na le liphello tse tšoenyang, e leng se etsang hore e be phekolo e ka 'nang ea e-ba teng bakeng sa mafu a ho tšoenyeha a kang lefu la ho tšoenyeha ka kakaretso le lefu la ho tšoenyeha ha sechaba.

Lisebelisoa

Tianeptine Hemisulfate Monohydrate ke lik'hemik'hale tse sebelisoang haholo tsa meriana likarolong tsa bongaka le tsa lipatlisiso.E le sethethefatsi se thibelang ho tepella maikutlo, se amohetsoe linaheng tse ngata bakeng sa ho phekola khatello ea maikutlo, matšoenyeho, mathata a maikutlo le mafu a mang a amanang le ona.Ho feta moo, Tianeptine Hemisulfate Monohydrate e 'nile ea ithutoa ka bokhoni ba eona ba ho phekola mafu a neurodegenerative a kang Alzheimer's, taolo ea bohloko le phekolo ea bokhoba ba tahi.

Lilemong tsa morao tjena, Tianeptine Hemisulfate Monohydrate e fumane botumo bo ntseng bo eketseha liphuputsong tsa bongaka, haholo-holo ho nts'etsopele ea lithethefatsi tse thibelang ho imeloa kelellong.Ka lithuto tse ngata tse tiisang litlamorao tsa eona tsa kalafo, menyetla ea ts'ebeliso ea eona e ntse e bonahala butle-butle.Tianeptine Hemisulfate Monohydrate e ka fetoha lithethefatsi tse sebetsang ka bongata bakeng sa ho phekola mafu a fapaneng a methapo nakong e tlang.

Ho feta moo, Tianeptine Hemisulfate Monohydrate e boetse e na le lisebelisoa tse ka sebelisoang likarolong tse ling.Phuputso ea morao tjena e bontšitse hore Tianeptine Hemisulfate Monohydrate e ka 'na ea e-ba le monyetla oa ho phekola mafu a neurofunctional ka mor'a lefu la stroke.Ho feta moo, liphuputso tse ling li fana ka maikutlo a hore Tianeptine Hemisulfate Monohydrate e ka ba molemo bakeng sa mafu a metabolic a kang botenya le lefu la tsoekere.


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