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sehlahisoa

Moetsi oa phofo ea Coluracetam Nomoro ea CAS: 135463-81-9 99% bohloeki ba bonyane bakeng sa metsoako ea tlatsetso

Tlhaloso e Khutšoanyane:

Coluracetam ke setho sa lelapa la racetam la metsoako ea nootropic 'me e boetse e tsejoa e le MKC-231. E ntlafalitsoe ke Kobe Pharmaceutical Company Japane ka sepheo sa ho phekola AD le mathata a kelello.


Qaqiso ea Sehlahisoa

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Video ea Sehlahisoa

Liparamente tsa Sehlahisoa

Lebitso la sehlahisoa

Coluracetam

Lebitso le leng

MKC-231;

2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide

Nomoro ea CAS

135463-81-9

Foromo ea limolek'hule

C19H23N3O3

Boima ba limolek'hule

341.4

Bohloeki

99.0%

Ponahalo

Phofo e tšoeu

Kopo

Lisebelisoa tse Tala tsa Tlatsetso ea Lijo

Selelekela sa sehlahisoa

Coluracetam, setho sa lelapa la racemate la metsoako ea nootropic, e tsejoang hape e le MKC-231, ke motsoako oa nootropic o nang le litlamorao tse ntlafatsang tsebo le tse sireletsang methapo ea kutlo. Coluracetam e sebetsa ka ho fetola tsamaiso ea cholinergic. Ho nahanoa hore e eketsa maemo a acetylcholine, neurotransmitter ea bohlokoa bokong e amanang haufi-ufi le mesebetsi ea ho ithuta le ea memori. Coluracetam e etsa sena ka ho eketsa palo le ts'ebetso ea li-transporter tsa choline uptake, ka hona e ntlafatsa ho lokolloa ha acetylcholine le ho ntlafatsa matšoao lipakeng tsa li-neuron. Lithuto tse ling tsa pele tsa liteko le tsa liphoofolo li bontša hore Coluracetam e na le litlamorao tse ka bang teng tsa tšireletso ea methapo le tse ntlafatsang tsebo. Lithuto tse ling li fumane hore Coluracetam e na le phello e itseng ea ntlafatso holim'a ho senyeha ha mohopolo mehlala ea AD.

Tšobotsi

(1) Bohloeki bo phahameng: Coluracetam e lokisoa ho sebelisoa mekhoa e tsoetseng pele ea ho ntša le ho etsa tlhahiso ho netefatsa bohloeki bo phahameng. Bohloeki bona bo phahameng bo thusa ho ntlafatsa ho fumaneha ha 'mele le ho fokotsa ho hlaha ha likarabelo tse mpe.
(2) Polokeho: Coluracetam e nkoa e sireletsehile bakeng sa batho. Palo e kholo ea lithuto e pakile hore e na le chefo e tlase le litla-morao tse fokolang ka har'a tekanyo e khothaletsoang.
(3) Botsitso: Litokisetso tsa Coluracetam li bontša botsitso bo botle 'me li ka boloka ts'ebetso ea tsona le katleho tlas'a maemo a fapaneng a tikoloho le maemo a polokelo. Botsitso bona bo netefatsa ts'ebetso e tsitsitseng le e tšepahalang ka nako e telele.

Likopo

Coluracetam hajoale e sebelisoa lits'ebetsong tse fapaneng 'me e bontša tšepiso e kholo ea bokamoso. E sebelisoa haholo-holo e le tlatsetso ea lijo e ntlafatsang kelello 'me e batloa ke batho ba batlang ho ntlafatsa mohopolo, ho tsepamisa mohopolo le bokhoni ba ho ithuta. Ho nahanoa hore bokhoni ba motsoako ona ba ho fetola tsamaiso ea cholinergic bo kenya letsoho liphellong tsa eona tse ntlafatsang kelello. Ho feta moo, lipatlisiso li bontša hore Coluracetam e ka ba le thepa e sireletsang methapo ea kutlo e ka thusang ho thibela ho fokotseha ha kelello ho amanang le botsofali le ho tšehetsa bophelo bo botle ba boko ka kakaretso.


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