lebanta_la_page

sehlahisoa

Moetsi oa phofo ea Amino Tadalafil Nomoro ea CAS: 385769-84-6 Bohloeki ba 98% bonyane bakeng sa metsoako ea tlatsetso

Tlhaloso e Khutšoanyane:

Amino Tadalafil ke motsoako o tšoanang le Tadalafil, 'me lihlopha tse ling tse sebetsang sebopehong sa eona li nkeloa sebaka ke lihlopha tsa amino.


Qaqiso ea Sehlahisoa

Li-tag tsa Sehlahisoa

Video ea Sehlahisoa

Liparamente tsa Sehlahisoa

Lebitso la sehlahisoa

Amino Tadalafil

Lebitso le leng

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A-Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dion e;(6R,12aR)-2-Amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione

Nomoro ea CAS

385769-84-6

Foromo ea limolek'hule

C21H18N4O4

Boima ba limolek'hule

390.39

Bohloeki

98.0%

Ponahalo

Phofo e tšoeu ho isa ho e tšoeu

Kopo

Lisebelisoa tse Tala tsa Tlatsetso ea Lijo

Selelekela sa sehlahisoa

Amino Tadalafil ke motsoako o mocha, o tswang ho tadalafil, o ntseng o tuma haholo lefapheng la ho se sebetse hantle ha thobalano (ED). E kopanya amino acid le tadalafil, e leng sethibela-mafu sa PDE5 se amohetsweng ke FDA se sebediswang haholoholo ho phekola ED. E sebetsa ka ho eketsa phallo ya madi ho ya botoneng, e leng se dumellang banna ho fihlella le ho boloka ho ema. Ka lehlakoreng le leng, di-amino acid di bapala karolo ya bohlokwa mesebetsing e fapaneng ya mmele, ho kenyeletswa le tlhahiso ya diprotheine, e leng dibopeho tsa kaho ya dinama le ditho. Motswako wa metswako ena e mmedi o reretswe ho ntlafatsa katleho ya Tadalafil ho phekoleng ED. Mme amino Tadalafil ke mofuta o ntlafetseng o nang le bokgoni bo makatsang, o ntlafatsang tshebetso le ho tenyetseha ha pele ho yona. Sebopeho sa yona sa dikhemikhale se ntse se tshwana le Tadalafil, empa ka ho kenngwa ha dihlopha tsa amino, e fumana dibopeho tse ikgethang tse e etsang hore e hlahelle lefatsheng la meriana. Jwalo ka tadalafil, Amino Tadalafil e sebetsa ka ho thibela phosphodiesterase 5 (PDE5), enzyme e ikarabellang bakeng sa ho qhaqha cyclic guanosine monophosphate (cGMP) mmeleng. cGMP ke motsoako oa tlhaho o khothalletsang ho phomola ha methapo ea mali, ka hona o eketsa phallo ea mali. Ka ho thibela PDE5, amino Tadalafil e netefatsa ho bokellana ha cGMP, ka hona e ntlafatsa ho ruruha ha methapo ea mali le ho ntlafatsa phallo ea mali. Ho feta moo, bafuputsi ba hlahlobile bokhoni ba eona ba ho thusa ho phekola benign prostatic hyperplasia (BPH) ka ho khothaletsa phallo ea mali ho ea ho prostate.

Tšobotsi

(1) Bohloeki bo phahameng: Amino Tadalafil e ka fumana dihlahiswa tse hlwekileng haholo ka mekgwa ya tlhahiso e hlwekileng. Bohloeki bo phahameng bo bolela ho fumaneha ha dihlahiswa hantle le dikarabelo tse fokolang tse mpe.

(2) Polokeho: Polokeho e phahameng, dikarabelo tse fokolang tse mpe.

(3) Botsitso: Amino Tadalafil e na le botsitso bo botle mme e ka boloka ts'ebetso le phello ea eona tlas'a maemo a fapaneng a tikoloho le maemo a polokelo.

Likopo

Amino Tadalafil ke sethibela-mafu sa PDE5 se nang le ditlamorao tse tshwanang tsa meriana le tadalafil. Ka ho kopanya di-amino acid le tadalafil, ho nahannwa hore amino Tadalafil e sebetsa hantle haholo ho phekoleng bothata ba ho se sebetse hantle ha botona kapa botšehali ho feta tadalafil feela. Di-amino acid di ka thusa ho ntlafatsa phallo ya madi le ho tshehetsa katleho yohle ya meriana. Ho feta moo, e ka ntlafatsa matshwao a ho se sebetse hantle ha botona kapa botšehali (ED) ka ho thibela mosebetsi wa enzyme ya PDE5 ho kgothaletsa phallo ya madi ho ya dithong tsa botona kapa tsa botshehadi. Ha e bapiswa le tadalafil, amino Tadalafil e sisinyeha butle mmeleng mme e ka hlahisa ditlamorao tse nkang nako e telele. Sena se fa amino Tadalafil bokgoni bo boholo ba ho phekola ED.


  • E fetileng:
  • E 'ngoe:

  • Ngola molaetsa oa hau mona 'me u o romelle ho rona