Moetsi oa phofo ea Sunifiram CAS No.: 314728-85-3 99% bohloeki min.bakeng sa lisebelisoa tsa tlatsetso
Lihlahisoa tsa lihlahisoa
Lebitso la sehlahisoa | Sunifiram |
Lebitso le leng | 1-(4-Benzoylpiperazin-1-yl)propan-1-one;1-Benzoyl-4-(1-oxopropyl) piperazine |
Nomoro ea CAS. | 314728-85-3 |
Mokhoa oa limolek'hule | C14H18N2O2 |
Boima ba molek'hule | 246.30 |
Bohloeki | 99.0% |
Ponahalo | phofo e tšoeu ea kristale |
Ho paka | 1kg/ mokotla |
Kopo | lithethefatsi tsa nootropic |
Kenyelletso ea sehlahisoa
Sunifiram ke AMPA receptor agonist e ntlafatsang pontšo ho tsoa ho li-receptor tsa AMPA bokong, tseo ka kakaretso ho nahanoang hore ke libapali tsa bohlokoa tse amanang le ho ithuta le mohopolo.Ka ho ntlafatsa ts'ebetso ea li-receptor tsa AMPA, ho nahanoa hore Sunifiram e ntlafatsa bokhoni ba boko ba ho ithuta le ho hopola, ha e ntse e ntlafatsa mohopolo le matla a kelello.Ho feta moo e sebetsa ka ho susumetsa ts'ebetso ea li-receptor tsa glutamate le ho eketsa tlhahiso le ho lokolloa ha "acetylcholine" ea "learning neurotransmitter".Sunifiram e sebetsa haholo-holo e le ntho ea ampa, e bolelang hore e tlamella li-receptor tsa mofuta oa AMPA bokong ka mor'a ho tšela mokoallo oa mali-boko.Sena se hlohlelletsa tlhahiso ea glutamate, neurotransmitter ea bohlokoa e bohlokoa ho synaptic plasticity, kapa bokhoni ba methapo ea kutlo ho arabela ho eketseha kapa ho fokotseha ha ts'ebetso.Maemo a glutamate a bohlokoa ka ho khetheha ho hippocampus, karolo ea boko e phethang karolo e kholo ho tsamaisa sebaka le ho theha mohopolo le ho boloka, 'me maemo a lekaneng a glutamate a bohlokoa bakeng sa matla a nako e telele, kapa ntlafatso e tšoarellang, ea matla a pontšo pakeng tsa li-neurone. bohlokoa haholo.Boholo ba bokhoni ba Sunifiram ba ho ntlafatsa kelello qetellong bo fihleloa ka ho eketsa matla a matšoao a methapo karolong ena ea boko.
Sebopeho
(1) Ho ntlafatsa ho ithuta le ho hopola, sunifiram e sebetsa e le nootropic e matla, e fana ka lintlafatso tse ka lekanyetsoang ka lebelo la ho ithuta, ho boloka mohopolo, le ho hopola.
(2) E ka ntlafatsa ho tsepamisa maikutlo, ho susumetsa le ho hlaka kelellong.
(3) Ho matlafatsa maikutlo le matla.
(4) Pono e ntlafetseng le temoho, ka tsela e itseng, li tla etsa hore li be le ponahalo e khanyang haholoanyane, li etse hore khanya le moriti li bonahale haholoanyane, ’me mebala e hlake haholoanyane.