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sehlahisoa

Moetsi oa phofo ea Sunifiram Nomoro ea CAS: 314728-85-3 Bohloeki ba 99% bonyane bakeng sa metsoako ea tlatsetso

Tlhaloso e Khutšoanyane:

Sunifiram ke agonist ea AMPA receptor e ntlafatsang matšoao a tsoang ho li-receptor tsa AMPA bokong, tseo ka kakaretso li nkoang e le libapali tsa bohlokoa tse amanang le ho ithuta le ho hopola.


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Lebitso la sehlahisoa

Sunifiram

Lebitso le leng

1-(4-Benzoylpiperazin-1-yl)propan-1-e le 'ngoe; 1-Benzoyl-4-(1-oxopropyl)piperazine

Nomoro ea CAS

314728-85-3

Foromo ea limolek'hule

C14H18N2O2

Boima ba limolek'hule

246.30

Bohloeki

99.0%

Ponahalo

phofo e tšoeu ea kristale

Ho paka

1kg/mokotla

Kopo

lithethefatsi tsa nootropic

Selelekela sa sehlahisoa

Sunifiram ke agonist ea AMPA receptor e ntlafatsang matshwao a lesedi ho li-receptor tsa AMPA bokong, tseo hangata ho nahanoang hore li phetha karolo ea bohlokoa ho ithuteng le ho hopoleng. Ka ho ntlafatsa ts'ebetso ea li-receptor tsa AMPA, Sunifiram ho nahanoa hore e ntlafatsa bokhoni ba boko ba ho ithuta le ho hopola, ha ka nako e ts'oanang e ntlafatsa ho tsepamisa mohopolo le matla a kelello. Ho feta moo, e sebetsa ka ho hlasimolla ts'ebetso ea li-receptor tsa glutamate le ho eketsa tlhahiso le ho lokolloa ha acetylcholine ea "learning neurotransmitter". Sunifiram e sebetsa haholo-holo e le ampa factor, ho bolelang hore e tlamahana le li-receptor tsa glutamate tsa mofuta oa AMPA bokong ka mor'a ho tšela mokoallo oa mali le boko. Sena se hlasimolla tlhahiso ea glutamate, neurotransmitter ea bohlokoa e bohlokoa bakeng sa plasticity ea synaptic, kapa bokhoni ba li-synapses tsa methapo ho arabela keketseho kapa phokotso ea ts'ebetso. Maemo a Glutamate a bohlokoa haholo ho hippocampus, karolo ea boko e bapalang karolo ea bohlokoa ho tsamaiseng sebaka, ho thehoeng ha memori le polokelo. Maemo a glutamate a lekaneng a bohlokoa bakeng sa ntlafatso ea nako e telele kapa ntlafatso e tšoarellang ea matšoao lipakeng tsa li-neuron. Matla a bohlokoa. Bongata ba matla a ho ntlafatsa tsebo a Sunifilaram qetellong a sebetsa ka ho eketsa matla a matšoao a methapo karolong ena ea boko.

Tšobotsi

(1) Bohloeki bo phahameng: Sunifiram e ka fumana dihlahiswa tse hlwekileng haholo ka mekgwa ya tlhahiso e hlwekileng. Bohloeki bo phahameng bo bolela ho fumaneha ha dikokwana-hloko ho betere le dikarabelo tse fokolang tse mpe.

(2) Polokeho: Sunifiram e pakiloe e sireletsehile bakeng sa 'mele oa motho.

(3) Botsitso: Sunifiram e na le botsitso bo botle mme e ka boloka ts'ebetso le phello ea eona tlas'a maemo a fapaneng a tikoloho le maemo a polokelo.

Likopo

Sunifiram ke sesebelisoa se ntlafatsang methapo ea kutlo, se fumanehang hape e le tlatsetso ea lijo, se nahanoang hore se ntlafatsa ts'ebetso ea kelello le ho ntlafatsa ho ithuta le mohopolo. E sebetsa ka ho sebetsana le li-receptor tsa AMPA bokong. AMPA ke neurotransmitter e amehang puisanong e potlakileng lipakeng tsa lisele tse tsamaisong ea methapo. E ntlafatsa haholo lebelo la ho ithuta, ho boloka mohopolo le ho hopola, hammoho le ho ntlafatsa ho tsepamisa mohopolo, khothatso le ho hlaka ha kelello.


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