Moetsi oa phofo ea Pramiracetam CAS No.: 68497-62-1 98% bohloeki min.bakeng sa lisebelisoa tsa tlatsetso
Lihlahisoa tsa lihlahisoa
Lebitso la sehlahisoa | Pramiracetam |
Lebitso le leng | Amacetam; N- [2-(Diisopropylamino) ethyl] -2-oxo-1-pyrrolidineacetamide;N-(2-(Bis(1-methylethyl)amino)ethyl) -2-oxo-1-pyrrolidineacetamide; NeupraMir; PraMistar; ReMen; Vinpotropil |
Nomoro ea CAS | 68497-62-1 |
Mokhoa oa limolek'hule | C14H27N3O2 |
Boima ba molek'hule | 269.38 |
Bohloeki | 99.0% |
Ponahalo | Phofo e tšoeu ea kristale |
Ho paka | 25kg/barrel |
Kopo | Nootropic |
Kenyelletso ea sehlahisoa
Pramiracetam ke sethethefatsi se ntlafatsang metabolism ea boko sa pyrrolidone, e leng moriana o bohareng oa methapo o ka ntlafatsang mohopolo le ho thibela ho lebala.E thehiloe ke Parke-Davis Pharmaceutical Company United States, Pramiracetam e na le bokhoni bo matla ba ho ntlafatsa ts'ebetso ea boko, ho ntlafatsa mohopolo le ho khothalletsa ho falimeha ha boko.Liteko tsa bongaka li pakile hore ts'ebetso ea eona ke makhetlo a 6-13 ho feta a piracetam (ho tsosolosoa ha cerebral).Ke makhetlo a 3-4 ho feta oxacetam le makhetlo a 1.25 ho feta aniracetam e ngata.Ka chefo e tlase le mamello e ntle, e ka sebelisoa bakeng sa meriana ea nako e telele ho ntlafatsa matšoao le ho liehisa 'dementia' ea Alzheimer.Ho loketse hore batho ba tsofetseng ba hlokomeloe le mathata a ho hopola, ho lebala botsofali bo botle, thibelo ea 'dementia' (lefu la Alzheimer's), ho ntlafatsa mohopolo.Pramiracetam e boetse e sebelisoa e le tlatsetso lihlahisoa tsa tlhokomelo ea bophelo bakeng sa mohaho oa 'mele le ho fokotseha ha methapo ea mali.
Sebopeho
Pramiracetam e sebetsa ka ho eketsa ho lokolloa ha neurotransmitter acetylcholine ho ntlafatsa ts'ebetso ea kelello bokong.E ka boela ea eketsa palo le khokahanyo ea methapo ea kutlo, ea khothalletsa kholo ea neuron le ho lokisa.Pramiracetam e ka boela ea eketsa lebelo la metabolism ea boko le ho eketsa phallo ea mali ea boko, kahoo e ntlafatsa phepelo ea oksijene le limatlafatsi bokong.Pramiracetam e sebelisoa haholo ho phekola mathata a kang ho senyeha ha kelello, ho lahleheloa ke mohopolo, ho se tsotelle le mathata a ho ithuta.E boetse e sebelisoa ho ntlafatsa ts'ebetso ea liatleletiki le ho fokotsa matšoao a ho tšoenyeha le ho tepella maikutlong.
Lisebelisoa
Pramiracetam ke moemeli ea matla oa nootropic eo e leng setho sa lelapa la lithethefatsi la racetam.Pramiracetam e ntlafatsa bofokoli ba kelello bo amanang le likotsi tse sithabetsang tsa boko.Hape, Pramiracetam ke inhibitor e khethehileng ea prolyl endopeptidase.Pramiracetam e phetha karolo ea bohlokoa thutong ea sebaka le mohopolong oa likhoto.E nkoa e le moemeli oa ho hopola mohopolo 'me e matla ho feta piracetam.